A 987306 | Tocris Bioscience 3640 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

A 987306

catalog :

3640

quantity :

10 mg (also 50 mg)

price :

261 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

3640

SKU :

3640/10

product name :

A 987306

description :

Potent and selective H4 antagonist

target :

Histamine H4 Receptor Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

327.42

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent histamine H4 receptor antagonist (pKi values are 8.24 and 8.47 in human and rat H4 receptors respectively). Displays 162-fold, 620-fold, and 1600-fold selectivity over human H3, H1 and H2 receptors. Blocks zymosan-induced neutrophil reflux and attenuates thermal hypersensitivity in vivo (ED50 = 42 mol/kg, ip).

catalog number base :

3640

product keywords :

potent selective H4 histamine histaminergic receptors antagonists A987306 Histamine H4 Receptors 3640,

extended description :

Potent and selective H4 antagonist

chemical name text :

( )-(7aR*,11aR*)-5,6,7a,8,9,10,11,11a-Octahydro-4-(1-piperazinyl)-benzofuran[2,3-h]quinazolin-2-amine

formula :

C 18 H 25 N 5 O

formula text :

C18H25N5O

cas num :

1082954-71-9

2020 USD :

255

2021 USD :

261 USD

storage :

Store at -20°C

more info or order :

Tocris Bioscience product webpage