CHR 2797 | Tocris Bioscience 3595 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

CHR 2797

catalog :

3595

quantity :

1 mg (also 10 mg)

price :

149 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

3595

SKU :

3595/1

product name :

CHR 2797

description :

Aminopeptidase inhibitor

target :

Aminopeptidase Inhibitors

category :

Small Molecules

unit size :

1 mg (also 10 mg)

purity :

98%

observed molecular weight :

406.48

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Aminopeptidase inhibitor (IC50 values are 100, 150, 220, 1000, 5000, 10000 and 30000 nM for LAP, PuSA, aminopeptidase N, aminopeptidase B, PILSAP, LTA4 hydrolase and MetAP2, respectively). Potently inhibits tumor cell proliferation in a variety of tumor cell lines in vitro and in vivo . Also inhibits neprilysin (IC50 = 900 nM). Exhibits antinociceptive activity and enhances the efficacy of Morphine (Cat. No. 5158) in the hot-plate and tail-flick assays, via an action on the peripheral nervous system.

catalog number base :

3595

product keywords :

aminopeptidases inhibitors inhibits proteases proteinases CHR2797 neprilysin neutral endopeptidase NEP Tosedostat Aminopeptidases 3595,

extended description :

Aminopeptidase inhibitor

chemical name text :

-[[(2R)-2-[(1S)-1-Hydroxy-2-(hydroxyamino)-2-oxoethyl]-4-methyl-1-oxopentyl]amino]-benzeneacetic acid cyclopently ester

formula :

C 21 H 30 N 2 O 6

formula text :

C21H30N2O6

cas num :

238750-77-1

2020 USD :

144

2021 USD :

149 USD

alt names :

Tosedostat

storage :

Store at -20°C

more info or order :

Tocris Bioscience product webpage