product summary
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company name :
Tocris Bioscience
product type :
chemical
product name :
GSK 0660
catalog :
3433/10
quantity :
10 mg (also 50 mg)
price :
269 USD
more info or order :
citations: 20
Reference |
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Smith D, Martinelli R, Besra G, Illarionov P, Szatmari I, Brazda P, et al. Identification and characterization of a novel anti-inflammatory lipid isolated from Mycobacterium vaccae, a soil-derived bacterium with immunoregulatory and stress resilience properties. Psychopharmacology (Berl). 2019;: pubmed publisher
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Qian G, Fan W, Ahlemeyer B, Karnati S, Baumgart Vogt E. Peroxisomes in Different Skeletal Cell Types during Intramembranous and Endochondral Ossification and Their Regulation during Osteoblast Differentiation by Distinct Peroxisome Proliferator-Activated Receptors. PLoS ONE. 2015;10:e0143439 pubmed publisher
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Savage S, McCollum G, Yang R, Penn J. RNA-seq identifies a role for the PPARβ/δ inverse agonist GSK0660 in the regulation of TNFα-induced cytokine signaling in retinal endothelial cells. Mol Vis. 2015;21:568-76 pubmed
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product information
brand :
Tocris, a Bio-Techne brand
catalog number base :
3433
SKU :
3433/10
product name :
GSK 0660
description :
Selective PPAR antagonist
target :
PPAR delta Receptor Inverse Agonists
unit size :
10 mg (also 50 mg)
category :
Small Molecules
purity :
99%
storage :
Store at +4°C
observed molecular weight :
418.49
url print :
?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules
details of functionality :
GSK 0660 is a selective PPAR antagonist (IC50 values are 0.155, 10 and 10 M at PPAR , PPAR and PPAR respectively). Exhibits inverse agonist effects when administered by itself.
product keywords :
Selective PPAR PPARdelta antagonists Peroxisome Proliferator-activating Receptors GSK0660 PPARdelta Receptors 3433,
extended description :
Selective PPAR antagonist
chemical name text :
3-[[[2-Methoxy-4-(phenylamino)phenyl]amino]sulfonyl]-2-thiophenecarboxylic acid methyl ester
formula :
C19H18N2O5S2
formula text :
C19H18N2O5S2
cas num :
1014691-61-2
USD :
266
USD 2025 :
269 USD
product details :
Selective PPAR antagonist
more info or order :
company information

Tocris Bioscience
The Watkins Building
Atlantic Road
Avonmouth, Bristol
BS11 9QD
Atlantic Road
Avonmouth, Bristol
BS11 9QD
info@bio-techne.com
https://www.tocris.com800-343-7475
headquarters: UK
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