JKC 363 | Tocris Bioscience 3426/500 product information

product summary

request information :

company name :

Tocris Bioscience

product type :

chemical

product name :

JKC 363

catalog :

3426/500

quantity :

500µg

price :

129 USD

more info or order :

Tocris Bioscience product webpage

product information

CHEMISTRY :

NCCCC[C@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)[C@@H]1CSSCCC(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC2=CNC=N2)C(=O)N[C@H](CC2=CC3=CC=CC=C3C=C2)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC2=CNC3=C2C=CC=C3)C(=O)NCC(=O)N1)C(=O)N[C@@H](CC(O)=O)C(N)=O

Cat Number :

3426/500

Product Name :

JKC 363

Cas Number :

[436083-30-6]

Unit Size :

500µg

Size :

500

Unit :

µg

USD :

129 USD

Primary Category :

7-TM Receptors

Secondary Category :

Peptide Receptors

Tertiary Category :

Melanocortin Receptors

Primary Action :

Potent and selective MC4 receptor antagonist

Biological Description :

Potent and selective melanocortin MC4 receptor antagonist (IC50 values are 0.5 and 44.9 nM at MC4 and MC3 respectively) that antagonizes the effects of α-MSH. Suppresses thyrotropin-releasing hormone (TRH) release, attenuates food intake and reduces formalin-induced pain in vivo.

Formula :

C69H91N19O16S2

Molwt :

1506.72

more info or order :

Tocris Bioscience product webpage