YM 202074 sesquifumarate | Tocris Bioscience 3413 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

YM 202074 sesquifumarate

catalog :

3413

quantity :

25 mg

price :

368 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

3413

SKU :

3413/25

product name :

YM 202074 sesquifumarate

description :

High affinity, selective mGlu1 antagonist

target :

Group I mGluR Antagonists

category :

Small Molecules

unit size :

25 mg

purity :

99%

observed molecular weight :

588.67

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

High affinity, selective metabotropic glutamate receptor type 1 (mGlu1) antagonist. Binds an allosteric site of the rat mGlu1 receptor with a Ki of 4.8 nM. Inhibits mGlu1-mediated inositol phosphates production (IC50 = 8.6 nM in rat cerebellar granule cells). Neuroprotective in vivo .

catalog number base :

3413

product keywords :

selective YM202074 YM 202074 sesquifumarate metabotropic glutamate receptors antagonists mGluR1 mGlu mGlu1 Group I Receptors Glutamate (Metabotropic) Group I Receptors 3413,

extended description :

High affinity, selective mGlu1 antagonist

chemical name text :

N-Cyclohexyl-6-[[N-(2-methoxyethyl)-N-methylamino]methyl]-N-methylthiazolo[3,2-a]benzoimidazole-2-carboxamide sesquifumarate

formula :

C 22 H 30 N 4 O 2 S.1.5C 4 H 4 O 4

formula text :

C22H30N4O2S.1.5C4H4O4

cas num :

299900-84-8

2020 USD :

360

2021 USD :

368 USD

storage :

Store at +4°C

more info or order :

Tocris Bioscience product webpage