VU 152100 | Tocris Bioscience 3383/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

VU 152100

catalog :

3383/10

quantity :

10 mg (also 50 mg)

price :

231 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris, a Bio-Techne Brand

catalog number base :

3383

SKU :

3383/10

product name :

VU 152100

Description :

Positive allosteric modulator of M4 receptors

target :

mAChR M4 Modulators

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

341.43

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

VU 152100 is a selective positive allosteric modulator of M4 muscarinic acetylcholine receptors (mAChRs) (EC50 = 380 nM). Induces 21-fold shift in ACh potency at M4 receptor. Displays no activity at other mAChR subtypes.

extended description :

Positive allosteric modulator of M4 receptors

chemical name text :

3-Amino-N-(4-methoxybenzyl)-4,6-dimethylthieno[2,3-b]pyridine carboxamide

formula :

C 18 H 19 N 3 O 2 S

formula text :

C18H19N3O2S

cas num :

409351-28-6

USD :

231 USD

product details :

Positive allosteric modulator of M4 receptors

alt names :

ML 108

storage :

Store at RT

more info or order :

Tocris Bioscience product webpage