SSR 146977 hydrochloride | Tocris Bioscience 3297/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

SSR 146977 hydrochloride

catalog :

3297/10

quantity :

10 mg (also 50 mg)

price :

331 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris, a Bio-Techne Brand

catalog number base :

3297

SKU :

3297/10

product name :

SSR 146977 hydrochloride

Description :

Potent and selective NK3 antagonist

target :

NK3 Receptor Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

658.11

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

SSR 146977 hydrochloride is a potent and selective NK3 receptor antagonist (Ki values are 0.26 and 19.3 nM in CHO cells expressing the human NK3 and NK2 receptor respectively). Also inhibits senktide -induced inositol monophosphate formation and intracellular calcium mobilization (IC50 = 10 nM).

extended description :

Potent and selective NK3 antagonist

chemical name text :

N1-[1-3-[(3R)-1-Benzoyl-3-(3-(3,4-dichlorophenyl)-3-piperidinyl]propyl]-4-phenyl-piperidinyl]-N,N-dimethylurea hydrochloride

formula :

C 35 H 42 Cl 2 N 4 O 2 .HCl

formula text :

C35H42Cl2N4O2.HCl

cas num :

264618-38-4

USD :

331 USD

product details :

Potent and selective NK3 antagonist

storage :

Store at +4°C

more info or order :

Tocris Bioscience product webpage