SB 452533 | Tocris Bioscience 3265 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

SB 452533

catalog :

3265

quantity :

10 mg (also 50 mg)

price :

163 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
Vijayvergiya V, Acharya S, Wilson S, Schmidt J. Measurement of Ensemble TRPV1 Ion Channel Currents Using Droplet Bilayers. PLoS ONE. 2015;10:e0141366 pubmed publisher

product information

brand :

Tocris

master code :

3265

SKU :

3265/10

product name :

SB 452533

description :

Potent TRPV1 antagonist

target :

TRPV Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

376.29

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent TRPV1 antagonist against capsaicin (pKb = 7.7), noxious heat and acid-mediated (pIC50 = 7.0) receptor activation (pKi = 6.22 at the recombinant hTRPV1 receptor). Exhibits analgesic properties.

catalog number base :

3265

product keywords :

SB452533 TRPV1 transient receptor potential channels antagonists vanilloid receptors analgesic analgaesic TRPV 3265,

extended description :

Potent TRPV1 antagonist

chemical name text :

N-(2-Bromophenyl)-N -[2-[ethyl(3-methylphenyl)amino]ethyl]-urea

formula :

C 18 H 22 BrN 3 O

formula text :

C18H22BrN3O

cas num :

459429-39-1

2020 USD :

163

2021 USD :

163 USD

storage :

Store at RT

more info or order :

Tocris Bioscience product webpage