SCH 221510 | Tocris Bioscience 3240/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

SCH 221510

catalog :

3240/10

quantity :

10 mg (also 50 mg)

price :

289 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
Wu Q, Liu L. ORL1 Activation Mediates a Novel ORL1 Receptor Agonist SCH221510 Analgesia in Neuropathic Pain in Rats. J Mol Neurosci. 2018;66:10-16 pubmed publisher

product information

brand :

Tocris, a Bio-Techne Brand

catalog number base :

3240

SKU :

3240/10

product name :

SCH 221510

Description :

Potent and selective NOP agonist

target :

NOP Receptor Agonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

99%

observed molecular weight :

397.55

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

SCH 221510 is a potent and selective nociceptin opioid receptor (NOP) agonist (EC50 values are 12, 693, 683 and 8071 nM, and Ki values are 0.3, 65, 131 and 2854 nM at NOP, -, - and -opioid receptors respectively). Exhibits anxiolytic-like activity at doses that have no effect on overt behaviors such as locomotion in vivo . Orally active.

extended description :

Potent and selective NOP agonist

chemical name text :

3-Endo-8-[bis(2-methylphenyl)methyl]-3-phenyl-8-azabicyclo[3.2.1]octan-3-ol

formula :

C 28 H 31 NO

formula text :

C28H31NO

cas num :

322473-89-2

USD :

289 USD

product details :

Potent and selective NOP agonist

storage :

Store at RT

more info or order :

Tocris Bioscience product webpage