Conantokin-R | Tocris Bioscience 3125/500 product information

product summary

request information :

company name :

Tocris Bioscience

product type :

chemical

product name :

Conantokin-R

catalog :

3125/500

quantity :

500µg

price :

265 USD

more info or order :

Tocris Bioscience product webpage

product information

CHEMISTRY :

[H]NCC(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(C(O)=O)C(O)=O)C(=O)N[C@@H](CC(C(O)=O)C(O)=O)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C(O)=O)C(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC(C(O)=O)C(O)=O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCCN)C(=O)NCC(=O)N[C@H]1CSSC[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC1=O)C(C)C)C(=O)N[C@@H](CC1=CC=C(O)C=C1)C(=O)N1CCC[C@H]1C(O)=O

Cat Number :

3125/500

Product Name :

Conantokin-R

Cas Number :

[202925-60-8]

Unit Size :

500µg

Size :

500

Unit :

µg

USD :

265 USD

Primary Category :

Ion Channels

Secondary Category :

Ligand-gated Ion Channels

Tertiary Category :

Glutamate (Ionotropic) Receptors

Primary Action :

Potent non-competitive NMDA receptor antagonist

Biological Description :

Potent, non-competitive NMDA receptor antagonist (IC50 = 93 nM) that has been suggested to have NR2 subunit selectivity. Inhibits inward currents evoked by NMDA in central nervous system neurons (IC50 = 350 nM) and exhibits broad anticonvulsant and antiparkinsonian activity in vivo at doses devoid of behavioral toxicity.

Formula :

C127H201N35O49S3

Molwt :

3098.4

more info or order :

Tocris Bioscience product webpage