XRP44X | Tocris Bioscience 3101/50 product information

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product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

XRP44X

catalog :

3101/50

quantity :

50 mg

price :

809 USD

product information

CHEMISTRY :

CC1=NN(C2=CC=CC=C2)C(C(N3CCN(C4=CC(Cl)=CC=C4)CC3)=O)=C1

Stock Reference :

3101/50

Cat Number :

3101

Product Name :

XRP44X

Cas Number :

[729605-21-4]

Unit Size :

50 mg

Size :

Unit :

USD :

809 USD

Primary Category :

Enzymes

Secondary Category :

GTPases

Tertiary Category :

Small Monomeric GTPases

Primary Action :

Ras-Net (Elk-3) pathway inhibitor; also microtubule depolymerization agent and angiogenesis inhibitor

Biological Description :

Ras-Net (Elk-3) pathway inhibitor (IC50 = 10 - 20 nM). Indirectly inhibits Net phosphorylation upstream of Erk1/2 activation. Mediates G2-M cell cycle arrest, suppresses growth of multiple cell types (IC50 ~ 2 nM), inhibits angiogenesis and acts as a microtubule depolymerizing agent in vitro.

Storage :

Store at RT

Formula :

C21H21ClN4O

Molwt :

380.87

Minimum Purity :

> 99%

Solubility :

Soluble to 100 mM in DMSO and to 50 mM in ethanol