L-651,582 | Tocris Bioscience 3086 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

L-651,582

catalog :

3086

quantity :

10 mg (also 50 mg)

price :

216 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

3086

SKU :

3086/10

product name :

L-651,582

description :

Non-selective Ca2+ channel blocker

target :

Voltage-gated Calcium Channel Blockers

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

424.67

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Orally active Ca2+ channel blocker; inhibits K+- and carbachol-stimulated Ca2+ influx (IC50 values are 500 and 935 nM respectively). Exhibits antiproliferative, antiangiogenic and antimetastatic activity in vivo and displays selectivity towards numerous mismatch repair-deficient tumor cell lines in vitro .

catalog number base :

3086

product keywords :

Ca2+ channel blockers Calcium CaV Channels voltage-gated voltage-dependent L651582 Carboxyamidotriazole Non-selective Cav Channels 3086, Voltage-gated calcium channel blocker, voltage gated calcium channel, high-voltage activated Ca2+ channel, high voltage gated ca2+ channel

extended description :

Non-selective Ca2+ channel blocker

chemical name text :

5-Amino-1-[[3,5-dichloro-4-(4-chlorobenzoyl)phenyl]methyl]-1H-1,2,3-triazole-4-carboxamide

formula :

C 17 H 12 Cl 3 N 5 O 2

formula text :

C17H12Cl3N5O2

cas num :

99519-84-3

2020 USD :

209

2021 USD :

216 USD

alt names :

Carboxyamidotriazole

storage :

Store at +4°C

more info or order :

Tocris Bioscience product webpage