LY 272015 hydrochloride | Tocris Bioscience 3077/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

LY 272015 hydrochloride

catalog :

3077/10

quantity :

10 mg (also 50 mg)

price :

272 USD

more info or order :

Tocris Bioscience product webpage

citations: 3

Reference
Watts S, Darios E, Seitz B, Thompson J. 5-HT is a potent relaxant in rat superior mesenteric veins. Pharmacol Res Perspect. 2015;3:e00103 pubmed publisher
Soll C, Riener M, Oberkofler C, Hellerbrand C, Wild P, DeOliveira M, et al. Expression of serotonin receptors in human hepatocellular cancer. Clin Cancer Res. 2012;18:5902-10 pubmed publisher
Niebert M, Vogelgesang S, Koch U, Bischoff A, Kron M, Bock N, et al. Expression and function of serotonin 2A and 2B receptors in the mammalian respiratory network. PLoS ONE. 2011;6:e21395 pubmed publisher

product information

brand :

Tocris, a Bio-Techne brand

catalog number base :

3077

SKU :

3077/10

product name :

LY 272015 hydrochloride

description :

High affinity 5-HT2B antagonist; orally active

target :

5-HT2B Receptor Antagonists

unit size :

10 mg (also 50 mg)

category :

Small Molecules

purity :

99%

storage :

Store at +4°C

observed molecular weight :

372.89

url print :

?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

LY 272015 hydrochloride is a high affinity 5-HT2B receptor antagonist that displays selectivity over 5-HT2A and 5-HT2C receptors (Ki values are 0.75, 21.63 and 28.7 nM for 5-HT2B, 5-HT2C and 5-HT2A receptors respectively). Orally active.

product keywords :

High affinity 5-HT2B antagonists orally active Serotonin Receptors LY272015 hydrochloride 5-HT2B Receptors 3077,

extended description :

High affinity 5-HT2B antagonist; orally active

chemical name text :

1-[(3,4-Dimethoxyphenyl)methy]-2,3,4,9-tetrahydro-6-methyl-1H-pyrido[3,4-b]indole hydrochloride

formula :

C21H24N2O2.HCl

formula text :

C21H24N2O2.HCl

cas num :

172895-15-7

USD :

269

USD 2025 :

272 USD

product details :

High affinity 5-HT2B antagonist; orally active

more info or order :

Tocris Bioscience product webpage