RO-3 | Tocris Bioscience 3052 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

RO-3

catalog :

3052

quantity :

10 mg

price :

141 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

3052

SKU :

3052/10

product name :

RO-3

description :

Selective P2X3 and P2X2/3 antagonist

target :

P2X Receptor Antagonists

category :

Small Molecules

unit size :

10 mg

purity :

98%

observed molecular weight :

302.37

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Selective homomeric P2X3 and heteromeric P2X2/3 receptor antagonist (pIC50 values are 7.0 and 5.9 respectively) that exhibits no activity at P2X1, P2X2, P2X4, P2X5 and P2X7 receptors (IC50 10 M). Attenuates nociceptive sensitivity in animal models of pain. Orally active and brain penetrant.

catalog number base :

3052

product keywords :

Selective P2X2 P2X2/3 antagonists Receptors Purinergic purinoceptors P2X Receptors 3052,

extended description :

Selective P2X3 and P2X2/3 antagonist

chemical name text :

5-[[4,5-Dimethoxy-2-(methylethyl)phenyl]methyl]-2,4-pyrimidinediamine

formula :

C 16 H 22 N 4 O 2

formula text :

C16H22N4O2

cas num :

1026582-88-6

2020 USD :

136

2021 USD :

141 USD

storage :

Store at RT

more info or order :

Tocris Bioscience product webpage