CI 1020 | Tocris Bioscience 2942 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

CI 1020

catalog :

2942

quantity :

1 mg (also 10 mg, 50 mg)

price :

100 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

2942

SKU :

2942/1

product name :

CI 1020

description :

Highly selective, orally active ETA antagonist

target :

Endothelin ETA Receptor Antagonists

category :

Small Molecules

unit size :

1 mg (also 10 mg, 50 mg)

purity :

98%

observed molecular weight :

506.5

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Highly selective, orally active, non-peptide endothelin-A receptor (ETA) antagonist (IC50 values are 0.3 and 480 nM for ETA and ETB receptors respectively). Antihypertensive; blocks ET-1-induced pressor responses following oral administration.

catalog number base :

2942

product keywords :

selective orally active ETA antagonists Receptors Endothelin CI1020 Pfizer PD156707 PD 156707 Endothelin ETA Receptors 2942,

extended description :

Highly selective, orally active ETA antagonist

chemical name text :

3-(1,3-Benzodioxol-5-yl)-5-hydroxy-5-(4-methoxyphenyl)-4-[(3,4,5-trimethoxyphenyl)methyl]-2(5H)-furanone

formula :

C 28 H 26 O 9

formula text :

C28H26O9

cas num :

162256-50-0

2020 USD :

2021 USD :

100 USD

alt names :

PD 156707

storage :

Store at -20°C

more info or order :

Tocris Bioscience product webpage