2789/10 | Tocris Bioscience 2789/10 product information

This webpage contains legacy information. The product is either no longer available from the supplier or has been delisted at Labome.

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

2789/10

catalog :

2789/10

quantity :

10 mg (also 50 mg)

price :

267 USD

citations: 2

Reference
Romei C, Bonifacino T, Milanese M, Usai C, Raiteri L. Colocalization of neurotransmitter transporters on the plasma membrane of the same nerve terminal may reflect cotransmission. Brain Res Bull. 2016;127:100-110 pubmed publisher
Debrouse L, Hurd B, Kiselycznyk C, Plitt A, Todaro A, Mishina M, et al. Probing the modulation of acute ethanol intoxication by pharmacological manipulation of the NMDAR glycine co-agonist site. Alcohol Clin Exp Res. 2013;37:223-33 pubmed publisher

product information

master code :

2789

SKU :

2789/10

product name :

NFPS

unit size :

10 mg (also 50 mg)

description :

Selective non-transportable GlyT1 inhibitor

target :

Glycine Transporter Inhibitors

category :

Small Molecules

purity :

98%

observed molecular weight :

393.45

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

NFPS is a selective, non-transportable inhibitor of GlyT1 which displays no activity at GABA or glutamate receptors (IC50 values are 2.8, 9.8 and 56000 nM for hGlyT1, rGlyT1 and rGlyT2 respectively). Enhances the amplitude of the NMDA component of glutamatergic EPSCs. . R-enantiomer also available.

top caption :

Selective non-transportable GlyT1 inhibitor

extended description :

Selective non-transportable GlyT1 inhibitor

chemical name text :

N-[3-([1,1-Biphenyl]-4-yloxy)-3-(4-fluorophenyl)propyl]-N-methylglycine

formula :

C24H24FNO3

formula text :

C24H24FNO3

cas num :

405225-21-0

USD :

267 USD

product details :

Selective non-transportable GlyT1 inhibitor

alt names :

( )-NFPS

storage :

Store at +4░C