L-365,260 | Tocris Bioscience 2767/10 product information

This webpage contains legacy information. The product is either no longer available from the supplier or has been delisted at Labome.

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

L-365,260

catalog :

2767/10

quantity :

10 mg (also 50 mg)

price :

253 USD

citations: 1

Reference
Wu W, Zhou H, He K, Pan X, Sugita Konishi Y, Watanabe M, et al. Role of cholecystokinin in anorexia induction following oral exposure to the 8-ketotrichothecenes deoxynivalenol, 15-acetyldeoxynivalenol, 3-acetyldeoxynivalenol, fusarenon X, and nivalenol. Toxicol Sci. 2014;138:278-89 pubmed publisher

product information

brand :

Tocris

master code :

2767

SKU :

2767/10

product name :

L-365,260

target :

CCK2 Receptor Antagonists

category :

Small Molecules

unit sizes :

10 mg (also 50 mg)

purity :

99%

observed molecular weight :

398.46

url print :

?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

L-365,260 is a selective cholecystokinin receptor 2 (CCK2) antagonist (IC50 values are 2 and 280 nM at CCK2 and CCK1 receptors respectively) that is inactive at a range of other receptors including opiate, muscarinic acetylcholine, - and adrenergic, histamine, angiotensin and bradykinin receptors.

extended description :

Selective CCK2 antagonist

chemical name text :

N-[(3R)-2,3-Dihydro-1-methyl-2-oxo-5-phenyl-1H-1,4-benzodiazepin-3-yl]-N -(3-methylphenyl)urea

formula :

C 24 H 22 N 4 O 2

formula text :

C24H22N4O2

cas num :

118101-09-0

USD :

253 USD

product details :

Selective CCK2 antagonist

storage :

Store at +4°C