PD 135158 | Tocris Bioscience 2608 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

PD 135158

catalog :

2608

quantity :

10 mg (also 50 mg)

price :

224 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

2608

SKU :

2608/10

product name :

PD 135158

description :

Potent and selective CCK2 antagonist

target :

CCK2 Receptor Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

616.76

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent and selective, nonpeptide CCK2 receptor antagonist (IC50 values are 2.8 and 1232 nM for CCK2 and CCK1 respectively) that displays negligible affinity at GABAA, benzodiazepine, substance P, neurotensin, opioid, bradykinin and 5-HT3 receptors (IC50 10 u M). Exhibits anxiolytic activity in elevated plus maze and social interaction tests and increases food intake in rats.

catalog number base :

2608

product keywords :

Potent selective CCK2 antagonists Cholecystokinin2 Receptors PD135158 CAM1028 CAM 1028 CCK2 Receptor 2608,

extended description :

Potent and selective CCK2 antagonist

chemical name text :

4-[[(1R)-2-[[(2R)-3-(1H-Indol-3-yl)-2-methyl-1-oxo-2-[[[[(1S,2R,4S)-1,7,7-trimethylbicyclo[2.2.1]hept-2-yl]oxy]carbonyl]amino]propyl]amino]-1-phenylethyl]amino]-4-oxobutanoic acid

formula :

C 35 H 44 N 4 O 6

formula text :

C35H44N4O6

cas num :

130285-87-9

2020 USD :

248

2021 USD :

224 USD

alt names :

CAM 1028

storage :

Store at +4°C

more info or order :

Tocris Bioscience product webpage