CI 988 | Tocris Bioscience 2607 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

CI 988

catalog :

2607

quantity :

10 mg (also 50 mg)

price :

320 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

2607

SKU :

2607/10

product name :

CI 988

description :

Potent and selective CCK2 antagonist

target :

CCK2 Receptor Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

99%

observed molecular weight :

614.73

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent and selective CCK2 (CCK-B) receptor antagonist that displays ~ 1600-fold selectivity over CCK1 receptors (IC50 values are 1.7 and 2717 nM for CCK2 and CCK1 respectively). Has negligible affinity at a range of other binding sites (IC50 10 u M). Exhibits anxiolytic activity following oral administration.

catalog number base :

2607

product keywords :

Potent selective CCK2 antagonists Cholecystokinin2 Receptors CI988 PD134308 PD 134308 CCK2 Receptor 2607,

extended description :

Potent and selective CCK2 antagonist

chemical name text :

4-[[(1R)-2-[[(2R)-3-(1H-indol-3-yl)-2-methyl-1-oxo-2-[[(tricyclo[3.3.1.13,7]dec-2-yloxy)carbonyl]amino]propyl]amino]-1-phenylethyl]amino]-4-oxobutanoic acid

formula :

C 35 H 42 N 4 O 6

formula text :

C35H42N4O6

cas num :

130332-27-3

2020 USD :

307

2021 USD :

320 USD

alt names :

PD 134308

storage :

Store at +4°C

more info or order :

Tocris Bioscience product webpage