2598/10 | Tocris Bioscience 2598/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

2598/10

catalog :

2598/10

quantity :

10 mg (also 50 mg)

price :

403 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
Wen Q, Yu G, Li Y, Yan L, Gong Z. Pharmacological mechanisms underlying the antinociceptive and tolerance effects of the 6,14-bridged oripavine compound 030418. Acta Pharmacol Sin. 2011;32:1215-24 pubmed publisher

product information

master code :

2598

SKU :

2598/10

product name :

(+/-)-J 113397

unit size :

10 mg (also 50 mg)

description :

Potent and selective NOP antagonist

target :

NOP Receptor Antagonists

category :

Small Molecules

purity :

98%

observed molecular weight :

399.57

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

( )-J 113397 is a potent and selective NOP receptor antagonist (IC50 values are 2.3, 1400, 2200 and 10000 nM for NOP, , u and -opioid receptors respectively). Inhibits nociceptin/orphanin FQ-induced hyperalgesia in the mouse tail-flick test.

top caption :

Potent and selective NOP antagonist

extended description :

Potent and selective NOP antagonist

chemical name text :

( )-1-[(3R*,4R*)-1-(Cyclooctylmethyl)-3-(hydroxymethyl)-4-piperidinyl]-3-ethyl-1,3-dihydro-2H-benzimidazol-2-one

formula :

C24H37N3O2

formula text :

C24H37N3O2

cas num :

217461-40-0

USD :

403 USD

product details :

Potent and selective NOP antagonist

storage :

Desiccate at RT

more info or order :

Tocris Bioscience product webpage