PD 166793 | Tocris Bioscience 2520 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

PD 166793

catalog :

2520

quantity :

10 mg (also 50 mg)

price :

151 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
Bencsik P, Kupai K, Gorbe A, Kenyeres E, Varga Z, Pálóczi J, et al. Development of Matrix Metalloproteinase-2 Inhibitors for Cardioprotection. Front Pharmacol. 2018;9:296 pubmed publisher

product information

brand :

Tocris

master code :

2520

SKU :

2520/10

product name :

PD 166793

description :

Broad spectrum MMP inhibitor

target :

Synthetic Metalloprotease Inhibitors

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

99%

observed molecular weight :

412.3

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Broad spectrum MMP inhibitor. Displays high affinity for MMP-2, -3 and -13 (IC50 values are 4, 7 and 8 nM respectively) and exhibits 750-fold selectivity over MMP-1, -7 and -9. Attenuates left ventricular remodelling and dysfunction in rat model of heart failure.

catalog number base :

2520

product keywords :

Broad spectrum MMP inhibitors inhibits Matrixins Matrix Metalloproteinase Metalloprotease Proteinases Proteases PD166793 Matrix Metalloprotease 2520,

extended description :

Broad spectrum MMP inhibitor

chemical name text :

N-[(4 -Bromo[1,1 -biphenyl]-4-yl)sulfonyl]-L-valine

formula :

C 17 H 18 BrNO 4 S

formula text :

C17H18BrNO4S

cas num :

199850-67-4

2020 USD :

145

2021 USD :

151 USD

storage :

Desiccate at +4°C

more info or order :

Tocris Bioscience product webpage