T 98475 | Tocris Bioscience 2519 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

T 98475

catalog :

2519

quantity :

1 mg

price :

221 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

2519

SKU :

2519/1

product name :

T 98475

description :

GnRH receptor antagonist

target :

Gonadotropin-Releasing Hormone Receptor (GnRH) Ant

category :

Small Molecules

unit size :

1 mg

purity :

98%

observed molecular weight :

657.77

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent, orally active and non-peptide gonadotropin-releasing hormone (GnRH, LHRH) receptor antagonist (IC50 values are 0.2, 4.0 and 60 nM for human, monkey and rat GnRH receptors respectively). Inhibits LH release in vitro (IC50 = 100 nM) and reduces plasma LH concentration in castrated male cynomolgus monkeys.

catalog number base :

2519

product keywords :

GnRH receptor antagonists Receptors Gonadotrophin-Releasing Hormone T98475 gonadotropin Gonadotrophin-Releasing Hormone Receptors 2519,

extended description :

GnRH receptor antagonist

chemical name text :

7-[(2,6-Difluorophenyl)methyl]-4,7-dihydro-2-[4-[(2-methyl-1-oxopropyl)amino]phenyl]-3-[[methyl(phenylmethyl)amino]methyl]-4-oxo-thieno[2,3-b]pyridine-5-carboxylic acid 1-methylethyl ester

formula :

C 37 H 37 F 2 N 3 O 4 S

formula text :

C37H37F2N3O4S

cas num :

199119-18-1

2020 USD :

216

2021 USD :

221 USD

storage :

Desiccate at +4°C

more info or order :

Tocris Bioscience product webpage