Trap 101 | Tocris Bioscience 2508 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

Trap 101

catalog :

2508

quantity :

10 mg

price :

148 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

2508

SKU :

2508/10

product name :

Trap 101

description :

Potent and selective NOP antagonist; active in vivo

target :

NOP Receptor Antagonists

category :

Small Molecules

unit size :

10 mg

purity :

98%

observed molecular weight :

434.02

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent and selective nociceptin/orphanin FQ (NOP) receptor antagonist (pA2 = 7.75). Displays selectivity for NOP receptors over classical opioid receptors (pKi values are 8.65, 6.60, 6.14 and 5 for NOP, -, -, and -opioid receptors respectively). Attenuates motor deficits in a rat model of Parkinson s Disease. Active in vivo .

catalog number base :

2508

product keywords :

Potent selective NOP antagonists Nociceptin Receptors ORL1 OP4 Opioid Trap101 Parkinsons disease antiparkinsons active in vivo NOP Receptors 2508,

extended description :

Potent and selective NOP antagonist; active in vivo

chemical name text :

1-[1-(Cyclooctylmethyl)-1,2,3,6-tetrahydro-5-(hydroxymethyl)-4-pyridinyl]-3-ethyl-1,3-dihydro-2H-benzimidazol-2-one hydrochloride

formula :

C 24 H 35 N 3 O 2 .HCl

formula text :

C24H35N3O2.HCl

cas num :

1216621-00-9

2020 USD :

185

2021 USD :

148 USD

storage :

Store at +4°C

more info or order :

Tocris Bioscience product webpage