Melperone hydrochloride | Tocris Bioscience 2495 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

Melperone hydrochloride

catalog :

2495

quantity :

10 mg (also 50 mg)

price :

81 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
Hacker K, Maas R, Kornhuber J, Fromm M, Zolk O. Substrate-Dependent Inhibition of the Human Organic Cation Transporter OCT2: A Comparison of Metformin with Experimental Substrates. PLoS ONE. 2015;10:e0136451 pubmed publisher

product information

brand :

Tocris

master code :

2495

SKU :

2495/10

product name :

Melperone hydrochloride

description :

5-HT2A antagonist; also D2 antagonist; neuroleptic

target :

5-HT2A Receptor Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

99%

observed molecular weight :

299.81

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Atypical neuroleptic; 5-HT2A/D2 receptor antagonist (Ki values are 120 and 180 nM respectively). Causes an increase in dopamine levels in the medial prefrontal cortex (mPFC) and nucleus accumbens and an increase in ACh in the mPFC. Also binds adrenergic 1 and 2 receptors (Ki values are 180 and 150 nM respectively).

catalog number base :

2495

product keywords :

5-HT2A/D2 receptor antagonists neuroleptic Serotonin Receptors Dopamine D2 dopaminergic 5-HT2A Receptors D2 Receptors 2495,

extended description :

5-HT2A antagonist; also D2 antagonist; neuroleptic

chemical name text :

1-(4-Fluorophenyl)-4-(4-methyl-1-piperidinyl)-1-butanone hydrochloride

formula :

C 16 H 22 FNO.HCl

formula text :

C16H22FNO.HCl

cas num :

1622-79-3

2020 USD :

2021 USD :

81 USD

storage :

Desiccate at RT

more info or order :

Tocris Bioscience product webpage