VUF 8430 dihydrobromide | Tocris Bioscience 2494 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

VUF 8430 dihydrobromide

catalog :

2494

quantity :

10 mg (also 50 mg)

price :

123 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
Martinel Lamas D, Cortina J, Ventura C, Sterle H, Valli E, Balestrasse K, et al. Enhancement of ionizing radiation response by histamine in vitro and in vivo in human breast cancer. Cancer Biol Ther. 2015;16:137-48 pubmed publisher

product information

brand :

Tocris

master code :

2494

SKU :

2494/10

product name :

VUF 8430 dihydrobromide

description :

Potent and high affinity H4 agonist

target :

Histamine H4 Receptor Agonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

observed molecular weight :

323.05

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

High affinity (pKi = 7.5), potent histamine H4 receptor full agonist (pEC50 = 7.3). Displays moderate affinity for H3 receptors (pKi = 6.0) and weak partial agonist activity at H2 receptors.

catalog number base :

2494

product keywords :

Potent high affinity H4 agonists Receptors Histamine histaminergic VUF8430 dihydrobromide Histamine H4 Receptors 2494,

extended description :

Potent and high affinity H4 agonist

chemical name text :

2-[(Aminoiminomethyl)amino]ethyl carbamimidothioic acid ester dihydrobromide

formula :

C 4 H 11 N 5 S.2HBr

formula text :

C4H11N5S.2HBr

cas num :

100130-32-3

2020 USD :

120

2021 USD :

123 USD

storage :

Desiccate at RT

more info or order :

Tocris Bioscience product webpage