VUF 8430 dihydrobromide | Tocris Bioscience 2494/10 product information

This webpage contains legacy information. The product is either no longer available from the supplier or has been delisted at Labome.

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

VUF 8430 dihydrobromide

catalog :

2494/10

quantity :

10 mg (also 50 mg)

price :

156 USD

citations: 1

Reference
Martinel Lamas D, Cortina J, Ventura C, Sterle H, Valli E, Balestrasse K, et al. Enhancement of ionizing radiation response by histamine in vitro and in vivo in human breast cancer. Cancer Biol Ther. 2015;16:137-48 pubmed publisher

product information

brand :

Tocris, a Bio-Techne brand

catalog number base :

2494

SKU :

2494/10

product name :

VUF 8430 dihydrobromide

description :

Potent and high affinity H4 agonist

target :

Histamine H4 Receptor Agonists

unit size :

10 mg (also 50 mg)

category :

Small Molecules

storage :

Desiccate at RT

observed molecular weight :

323.05

url print :

?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

VUF 8430 dihydrobromide is a high affinity (pKi = 7.5), potent histamine H4 receptor full agonist (pEC50 = 7.3). Displays moderate affinity for H3 receptors (pKi = 6.0) and weak partial agonist activity at H2 receptors.

product keywords :

Potent high affinity H4 agonists Receptors Histamine histaminergic VUF8430 dihydrobromide Histamine H4 Receptors 2494,

extended description :

Potent and high affinity H4 agonist

chemical name text :

2-[(Aminoiminomethyl)amino]ethyl carbamimidothioic acid ester dihydrobromide

formula :

C4H11N5S.2HBr

formula text :

C4H11N5S.2HBr

cas num :

100130-32-3

USD :

154

USD 2025 :

156 USD

product details :

Potent and high affinity H4 agonist