GT 2016 | Tocris Bioscience 2419 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

GT 2016

catalog :

2419

quantity :

10 mg (also 50 mg)

price :

130 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

2419

SKU :

2419/10

product name :

GT 2016

description :

Selective H3 antagonist

target :

Histamine H3 Receptor Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

317.47

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

High affinity H3 receptor antagonist (Ki = 43.8 nM). Displays selectivity against H1 and H2 receptors (IC50 10 M). Increases the release of histamine in the cerebral cortex. Displays no activity at histamine methyltransferase in vitro at concentrations up to 3 M. Brain penetrant.

catalog number base :

2419

product keywords :

GT2016 histamine h3 antagonists histaminergic selective brain penetrant centrally active Histamine H3 Receptors 2419,

extended description :

Selective H3 antagonist

chemical name text :

5-Cyclohexyl-1-[4-(1H-imidazol-5-yl)-1-piperidinyl]-1-pentanone

formula :

C 19 H 31 N 3 O

formula text :

C19H31N3O

cas num :

152241-24-2

2020 USD :

162

2021 USD :

130 USD

storage :

Store at -20°C

more info or order :

Tocris Bioscience product webpage