Gavestinel | Tocris Bioscience 2348 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

Gavestinel

catalog :

2348

quantity :

10 mg (also 50 mg)

price :

183 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

2348

SKU :

2348/10

product name :

Gavestinel

description :

Potent and selective NMDA antagonist; acts at the glycine site

target :

NMDA Receptor Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

397.19

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Highly potent and selective non-competitive antagonist acting at the strychnine-insensitive glycine binding site of the NMDA receptor-channel complex (Kd = 0.8 nM). Displays 1000-fold selectivity over NMDA, AMPA and kainate binding sites. Orally bioavailable and active in vivo .

catalog number base :

2348

product keywords :

Potent selective glycine site antagonists Orally available active vivo Glutamate NMDA Receptors N-Methyl-D-Aspartate iGluR Ionotropic GV150526A GlaxoSmithKline GSK GV 150526A NMDA Receptors 2348,

extended description :

Potent and selective NMDA antagonist; acts at the glycine site

chemical name text :

4,6-Dichloro-3-[(1E)-3-oxo-3-(phenylamino)-1-propenyl]-1H-indole-2-carboxylic acid sodium salt

formula :

C 18 H 11 Cl 2 N 2 O 3 Na

formula text :

C18H11Cl2N2O3Na

cas num :

153436-38-5

2020 USD :

179

2021 USD :

183 USD

alt names :

GV 150526A

storage :

Desiccate at RT

more info or order :

Tocris Bioscience product webpage