CGH 2466 dihydrochloride | Tocris Bioscience 2344 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

CGH 2466 dihydrochloride

catalog :

2344

quantity :

10 mg (also 50 mg)

price :

152 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
Wakisaka N, Miyasaka N, Koide T, Masuda M, Hiraki Kajiyama T, Yoshihara Y. An Adenosine Receptor for Olfaction in Fish. Curr Biol. 2017;27:1437-1447.e4 pubmed publisher

product information

brand :

Tocris

master code :

2344

SKU :

2344/10

product name :

CGH 2466 dihydrochloride

description :

A1, A2B and A3 antagonist and inhibitor of p38 MAPK and PDE4

target :

Non-selective Adenosine Receptor Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

99%

observed molecular weight :

395.13

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Adenosine A1, A2B and A3 receptor antagonist (IC50 values are 19, 21, and 80 nM respectively). Also inhibits p38 MAPK (IC50 = 187 - 400 nM) and phosphodiesterase type 4D (IC50 = 22 nM). Displays potent anti-inflammatory effects in vitro and in vivo . Potentially useful for asthma and chronic obstructive pulmonary disease (COPD) research.

catalog number base :

2344

product keywords :

A1 A2B A3 antagonists inhibitors inhibits p38 MAPK PDE4 Anti-inflammatory agent adenosines receptor Non-Selective Receptors Phosphodiesterases CGH2466 dihydrochloride Non-selective Adenosine Phosphodiesterases 2344,

extended description :

A1, A2B and A3 antagonist and inhibitor of p38 MAPK and PDE4

chemical name text :

4-(3,4-Dichlorophenyl)-5-(4-pyridinyl)-2-thiazolamine dihydrochloride

formula :

C 14 H 9 N 3 SCl 2 .2HCl

formula text :

C14H9N3SCl2.2HCl

cas num :

1177618-54-0

2020 USD :

152

2021 USD :

152 USD

storage :

Desiccate at +4°C

more info or order :

Tocris Bioscience product webpage