4-Methylhistamine dihydrochloride | Tocris Bioscience 2342 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

4-Methylhistamine dihydrochloride

catalog :

2342

quantity :

10 mg (also 50 mg)

price :

216 USD

more info or order :

Tocris Bioscience product webpage

citations: 4

Reference
Kim B, Kwon Y, Kim E, So I. Effects of histamine on cultured interstitial cells of cajal in murine small intestine. Korean J Physiol Pharmacol. 2013;17:149-56 pubmed publisher
Desmadryl G, Gaboyard Niay S, Brugeaud A, Travo C, Broussy A, Saleur A, et al. Histamine H4 receptor antagonists as potent modulators of mammalian vestibular primary neuron excitability. Br J Pharmacol. 2012;167:905-16 pubmed publisher
Connelly W, Shenton F, Lethbridge N, Leurs R, Waldvogel H, Faull R, et al. The histamine H4 receptor is functionally expressed on neurons in the mammalian CNS. Br J Pharmacol. 2009;157:55-63 pubmed publisher
Holden N, Gong W, King E, Kaur M, Giembycz M, Newton R. Potentiation of NF-kappaB-dependent transcription and inflammatory mediator release by histamine in human airway epithelial cells. Br J Pharmacol. 2007;152:891-902 pubmed

product information

brand :

Tocris

master code :

2342

SKU :

2342/10

product name :

4-Methylhistamine dihydrochloride

description :

Selective, high affinity H4 agonist

target :

Histamine H4 Receptor Agonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

observed molecular weight :

198.09

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent, high affinity H4 receptor agonist (Ki = 7 nM) that displays 100-fold selectivity over other human histamine receptor subtypes.

catalog number base :

2342

product keywords :

Selective high affinity H4 agonists Receptors Histamine histaminergic Histamine H4 Receptors 2342,

extended description :

Selective, high affinity H4 agonist

chemical name text :

5-(2-Aminoethyl)-4-methylimidazole dihydrochloride

formula :

C 6 H 11 N 3 .2HCl

formula text :

C6H11N3.2HCl

cas num :

36376-47-3

2020 USD :

207

2021 USD :

216 USD

storage :

Desiccate at RT

more info or order :

Tocris Bioscience product webpage