Raloxifene hydrochloride | Tocris Bioscience 2280 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

Raloxifene hydrochloride

catalog :

2280

quantity :

50 mg

price :

95 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
Nicholson T, Moses M, Uchtmann K, Keil K, Bjorling D, Vezina C, et al. Estrogen receptor-Î± is a key mediator and therapeutic target for bladder complications of benign prostatic hyperplasia. J Urol. 2015;193:722-9 pubmed publisher

product information

brand :

Tocris

master code :

2280

SKU :

2280/50

product name :

Raloxifene hydrochloride

description :

Selective estrogen receptor modulator (SERM)

target :

Estrogen and Related Receptor Modulators

category :

Small Molecules

unit size :

50 mg

purity :

98%

observed molecular weight :

510.04

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Selective estrogen receptor modulator (SERM) that binds to ER and ER , and tissue-dependently activates or blocks estrogen-induced transcription. Acts as an antiestrogen in breast and uterine tissue, but displays estrogen agonist activity in bone. In D12 rat hypothalamic cells, inhibits progesterone receptor induction by estrogen with an IC50 of 1 nM.

catalog number base :

2280

product keywords :

Selective estrogen receptor modulators SERM ER Estrogen Receptors LY139481 amino acid transporter 2 ASCT2 LY 139481 Keoxifene Estrogen and Related Receptors 2280,

extended description :

Selective estrogen receptor modulator (SERM)

chemical name text :

[6-Hydroxy-2-(4-hydroxyphenyl)benzo[b]thien-3-yl][4-[2-(1-piperidinyl)ethoxy]phenyl]-methanone hydrochloride

formula :

C 28 H 27 NO 4 S.HCl

formula text :

C28H27NO4S.HCl

cas num :

82640-04-8

2020 USD :

2021 USD :

95 USD

alt names :

LY 139481, Keoxifene

storage :

Desiccate at +4°C

more info or order :

Tocris Bioscience product webpage