LY 255283 | Tocris Bioscience 2208 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

LY 255283

catalog :

2208

quantity :

10 mg (also 50 mg)

price :

185 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
Cabral M, MartÃn Venegas R, Moreno J. Leukotriene D4-induced Caco-2 cell proliferation is mediated by prostaglandin E2 synthesis. Physiol Rep. 2015;3: pubmed publisher

product information

brand :

Tocris

master code :

2208

SKU :

2208/10

product name :

LY 255283

description :

Selective, competitive BLT2 receptor antagonist

target :

Leukotriene and Related Receptor Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

360.46

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Selective, competitive antagonist of BLT2 receptors (IC50 values are ~ 1 and 10 u M at human recombinant BLT2 and BLT1 receptors respectively). Inhibits LTB4-induced contraction of lung parenchyma (pA2 = 7.2), and reduces LTB4-mediated airway obstruction in guinea pigs following i.v. and oral administration.

catalog number base :

2208

product keywords :

Selective competitive BLT2 receptor antagonists CysLT1 Receptors CysLT2 BLT1 OXE Oxoeicosanoid receptors LTD4 LTE4 leukotrienes eicosanoids LY255283 Leukotriene and Related Receptors 2208,

extended description :

Selective, competitive BLT2 receptor antagonist

chemical name text :

1-[5-Ethyl-2-hydroxy-4-[[6-methyl-6-(1H-tetrazol-5-yl)heptyl]oxy]phenyl]ethanone

formula :

C 19 H 28 N 4 O 3

formula text :

C19H28N4O3

cas num :

117690-79-6

2020 USD :

179

2021 USD :

185 USD

storage :

Store at +4°C

more info or order :

Tocris Bioscience product webpage