NS 3763 | Tocris Bioscience 2187 product information

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product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

NS 3763

catalog :

2187

quantity :

10 mg (also 50 mg)

price :

164 USD

product information

brand :

Tocris

master code :

2187

SKU :

2187/10

product name :

NS 3763

description :

GluK1 selective and non-competitive kainate antagonist

target :

Kainate Receptor Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

404.38

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Selective non-competitive kainate receptor antagonist; displays selectivity for GluK1 (formerly GLUK5) subunit-containing receptors (IC50 values are 1.6 and 30 M for homomeric GluK1 (formerly GLUK5) and GluK2 (formerly GLUK6) receptors respectively). Has minimal activity at AMPA and NMDA receptors (IC50 30 M). . Please refer to IUPHAR Guide to Pharmacology for the most recent naming conventions .

catalog number base :

2187

product keywords :

Selective non-competitive kainate antagonists selective GLUK5 Glutamate Kainate Receptors iGluR Ionotropic NS3763 GluK1 Kainate Receptors 2187,

extended description :

GluK1 selective and non-competitive kainate antagonist

chemical name text :

4,6-Bis(benzoylamino)-1,3-benzenedicarboxylic acid

formula :

C 22 H 16 N 2 O 6

formula text :

C22H16N2O6

cas num :

70553-45-6

2020 USD :

160

2021 USD :

164 USD

storage :

Store at RT