(+/-)-McN 5652 | Tocris Bioscience 2148 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

(+/-)-McN 5652

catalog :

2148

quantity :

10 mg (also 50 mg)

price :

95 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

2148

SKU :

2148/10

product name :

(+/-)-McN 5652

description :

Potent, orally active 5-HT uptake inhibitor; also inhibits noradrenalin and dopamine uptake in vitro

target :

5-HT Transporter Inhibitors

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

295.44

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent, high affinity serotonin re-uptake inhibitor; selective in vivo . Displays moderate selectivity over noradrenalin and dopamine re-uptake in vitro (Ki values are 0.68, 2.9 and 36.8 nM for inhibition of serotonin, noradrenalin and dopamine uptake respectively in rat brain synaptosomes). Potently potentiates 5-HT-induced effects in vivo following oral administration. Biological activity resides predominantly in the (+)-enantiomer.

catalog number base :

2148

product keywords :

Potent orally active 5-HT reuptake inhibits inhibitors Transporters Monoamine Neurotransmitter Serotonin SERT 5-Hydroxytryptamine (?)-McN5652 McN5652Z McN 5652-Z 5-HT Transporters Adrenergic Transporters Dopamine Transporters 2148,

extended description :

Potent, orally active 5-HT uptake inhibitor; also inhibits noradrenalin and dopamine uptake in vitro

chemical name text :

(6R,10bS)-rel-1,2,3,5,6,10b-Hexahydro-6-[4-(methylthio)phenyl]-pyrrolo[2,1-a]isoquinoline

formula :

C 19 H 21 NS

formula text :

C19H21NS

cas num :

96795-89-0

2020 USD :

2021 USD :

95 USD

alt names :

McN 5652-Z

storage :

Store at -20°C

more info or order :

Tocris Bioscience product webpage