This webpage contains legacy information. The product is either no longer available from the supplier or has been delisted at Labome.
product summary
company name :
Tocris Bioscience
product type :
chemical
product name :
Cinalukast
catalog :
2025/10
quantity :
10 mg (also 50 mg)
price :
162 USD
citations: 1
Reference
Wright P, McCoull D, Walsh Y, Large J, Hadrys B, Gaurilcikaite E, et al. Pranlukast is a novel small molecule activator of the two-pore domain potassium channel TREK2. Biochem Biophys Res Commun. 2019;520:35-40 pubmed publisher
product information
brand :
Tocris
SKU :
2025/10
product name :
Cinalukast
unit sizes :
10 mg (also 50 mg)
description :
Potent, selective CysLT1 (LTD4) antagonist; orally active
target :
Leukotriene and Related Receptor Antagonists
category :
Small Molecules
purity :
98%
observed molecular weight :
412.55
details of functionality :
Potent, selective CysLT1 (LTD4) leukotriene receptor antagonist (IC50 = 6.4 nM). Inhibits LTD4-induced bronchoconstriction in guinea pigs when administered intravenously, orally or by aerosol.
catalog number base :
2025
extended description :
Potent, selective CysLT1 (LTD4) antagonist; orally active
chemical name text :
4-[[3-[(1E)-2-(4-Cyclobutyl-2-thiazolyl)ethenyl]phenyl]amino]-2,2-diethyl-4-oxobutanoic acid
formula :
C 23 H 28 N 2 O 3 S
formula text :
C23H28N2O3S
cas num :
128312-51-6
USD :
162 USD
product details :
Potent, selective CysLT1 (LTD4) antagonist; orally active
alt names :
Ro 24-5913
storage :
Desiccate at -20°C
company information
Tocris Bioscience
The Watkins Building
Atlantic Road
Avonmouth, Bristol
BS11 9QD
info@bio-techne.com
https://www.tocris.com
800-343-7475
headquarters: UK