product summary
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company name :
Tocris Bioscience
product type :
chemical
product name :
L-817,818
catalog :
1980/10
quantity :
10 mg
price :
398 USD
more info or order :
Tocris Bioscience product webpage
product information
brand :
Tocris, a Bio-Techne brand
catalog number base :
1980
SKU :
1980/10
product name :
L-817,818
description :
Potent and selective sst5 agonist
target :
Somatostatin Receptor Agonists
unit size :
10 mg
category :
Small Molecules
purity :
99%
storage :
Store at -20°C
observed molecular weight :
536.67
url print :
?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules
details of functionality :
L-817,818 is a potent and selective somatostatin sst5 receptor agonist. Ki values are 0.4, 3.3, 52, 64 and 82 nM for cloned human sst5, sst1, sst2, sst3 and sst4 receptors respectively. Inhibits growth hormone release from rat pituitary cells (EC50 = 3.1 nM) and insulin release from mouse pancreatic islets (EC50 = 0.3 nM) in vitro .
product keywords :
Potent selective sst5 agonists Receptors Somatostatin L817818 Somatostatin Receptors 1980,
extended description :
Potent and selective sst5 agonist
chemical name text :
N2-[[2-(2-Naphthalenyl)-1H-benz[g]indol-3-yl]acetyl-D-lysine (2S)-2-aminopropyl ester
formula :
C33H36N4O3
formula text :
C33H36N4O3
cas num :
217480-27-8
USD :
394
USD 2025 :
398 USD
product details :
Potent and selective sst5 agonist
more info or order :
Tocris Bioscience product webpage
company information
Tocris Bioscience
The Watkins Building
Atlantic Road
Avonmouth, Bristol
BS11 9QD
info@bio-techne.com
https://www.tocris.com
800-343-7475
headquarters: UK