L-803,087 trifluoroacetate | Tocris Bioscience 1979/10 product information

This webpage contains legacy information. The product is either no longer available from the supplier or has been delisted at Labome.

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

L-803,087 trifluoroacetate

catalog :

1979/10

quantity :

10 mg

price :

384 USD

product information

brand :

Tocris

master code :

1979

SKU :

1979/10

product name :

L-803,087 trifluoroacetate

description :

Potent and selective sst4 agonist

target :

Somatostatin Receptor Agonists

category :

Small Molecules

unit sizes :

10 mg

purity :

97%

observed molecular weight :

599.56

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

L-803,087 trifluoroacetate is a potent and selective somatostatin sst4 receptor agonist. Ki values are 0.7, 199, 4720, 1280 and 3880 nM for cloned human sst4, sst1, sst2, sst3 and sst5 receptors respectively. Facilitates AMPA-mediated hippocampal synaptic responses in vitro and increases kainate-induced seizures in mice in vivo .

extended description :

Potent and selective sst4 agonist

chemical name text :

N2-[4-(5,7-Difluoro-2-phenyl-1H-indol-3-yl)-1-oxobutyl]-L-arginine methyl ester trifluoroacetate

formula :

C 25 H 29 F 2 N 5 O 3 .CF 3 CO 2 H

formula text :

C25H29F2N5O3.CF3CO2H

cas num :

1786412-46-1

USD :

384 USD

product details :

Potent and selective sst4 agonist

storage :

Store at -20°C