HS 024 | Tocris Bioscience 1832 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

HS 024

catalog :

1832

quantity :

1 mg

price :

349 USD

more info or order :

Tocris Bioscience product webpage

citations: 2

Reference
Nepomuceno D, Kuei C, Dvorak C, Lovenberg T, Liu C, Bonaventure P. Re-evaluation of Adrenocorticotropic Hormone and Melanocyte Stimulating Hormone Activation of GPR139 in Vitro. Front Pharmacol. 2018;9:157 pubmed publisher
Simamura E, Arikawa T, Ikeda T, Shimada H, Shoji H, Masuta H, et al. Melanocortins contribute to sequential differentiation and enucleation of human erythroblasts via melanocortin receptors 1, 2 and 5. PLoS ONE. 2015;10:e0123232 pubmed publisher

product information

brand :

Tocris

master code :

1832

SKU :

1832/1

product name :

HS 024

description :

Highly potent MC4 receptor antagonist

target :

Melanocortin Receptor Antagonists

category :

Peptides

unit size :

1 mg

observed molecular weight :

1266.5

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=peptides

details of functionality :

Highly potent melanocortin MC4 receptor antagonist (Ki values are 0.29, 18.6, 5.45 and 3.29 nM for cloned human MC4, MC1, MC3 and MC5 receptors respectively). Increases food intake, and blocks -MSH- and MTII-induced hypotension and bradycardia in rats, following central administration in vivo .

catalog number base :

1832

product keywords :

potent MC4R receptor antagonists Receptors Melanocortin HS024 Melanocortin Receptors 1832,

extended description :

Highly potent MC4 receptor antagonist

formula :

C 58 H 79 N 19 O 10 S 2

formula text :

C58H79N19O10S2

cas num :

212370-59-7

2020 USD :

335

2021 USD :

349 USD

storage :

Desiccate at -20°C

more info or order :

Tocris Bioscience product webpage