HS 024 | Tocris Bioscience 1832/1 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

HS 024

catalog :

1832/1

quantity :

1 mg

price :

439 USD

more info or order :

Tocris Bioscience product webpage

citations: 2

Reference
Nepomuceno D, Kuei C, Dvorak C, Lovenberg T, Liu C, Bonaventure P. Re-evaluation of Adrenocorticotropic Hormone and Melanocyte Stimulating Hormone Activation of GPR139 in Vitro. Front Pharmacol. 2018;9:157 pubmed publisher
Simamura E, Arikawa T, Ikeda T, Shimada H, Shoji H, Masuta H, et al. Melanocortins contribute to sequential differentiation and enucleation of human erythroblasts via melanocortin receptors 1, 2 and 5. PLoS ONE. 2015;10:e0123232 pubmed publisher

product information

brand :

Tocris

catalog number base :

1832

SKU :

1832/1

product name :

HS 024

units size :

1 mg

description :

Highly potent MC4 receptor antagonist

target :

Melanocortin Receptor Antagonists

category :

Peptides

purity :

95%

observed molecular weight :

1266.5

url print :

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details of functionality :

HS 024 is a highly potent melanocortin MC4 receptor antagonist (Ki values are 0.29, 18.6, 5.45 and 3.29 nM for cloned human MC4, MC1, MC3 and MC5 receptors respectively). Increases food intake, and blocks -MSH- and MTII-induced hypotension and bradycardia in rats, following central administration in vivo .

top caption :

Highly potent MC4 receptor antagonist

extended description :

Highly potent MC4 receptor antagonist

formula :

C58H79N19O10S2

formula text :

C58H79N19O10S2

cas num :

212370-59-7

USD :

439 USD

product details :

Highly potent MC4 receptor antagonist

storage :

Store at -20Â°C

more info or order :

Tocris Bioscience product webpage