OMDM-2 | Tocris Bioscience 1797 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

OMDM-2

catalog :

1797

quantity :

25 mg

price :

253 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
Batkai S, Pacher P, Osei Hyiaman D, Radaeva S, Liu J, Harvey White J, et al. Endocannabinoids acting at cannabinoid-1 receptors regulate cardiovascular function in hypertension. Circulation. 2004;110:1996-2002 pubmed

product information

brand :

Tocris

master code :

1797

SKU :

1797/25

product name :

OMDM-2

description :

Potent inhibitor of anandamide uptake

target :

Cannabinoid Transporter Inhibitors

category :

Small Molecules

unit size :

25 mg

purity :

99%

observed molecular weight :

431.66

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Metabolically stable inhibitor of anandamide cellular uptake (Ki = 3 u M). Displays relatively low affinity for CB1 and CB2 receptors (Ki values are 5.1 and 10 u M) and for vanilloid VR1 receptors (EC50 = 10 u M). FABP inhibitor. Has minimal activity against FAAH (Ki 50 u M). Active in vivo .

catalog number base :

1797

product keywords :

Potent inhibitors inhibits anandamide reuptake AMT Transporters cannabinoids Monoamine Neurotransmitter FABPs FABP fatty acid binding proteins Cannabinoid Transporters Fatty Acid Binding Proteins 1797,

extended description :

Potent inhibitor of anandamide uptake

chemical name text :

(9Z)-N-[1-((R)-4-Hydroxbenzyl)-2-hydroxyethyl]-9-octadecenamide

formula :

C 27 H 45 NO 3

formula text :

C27H45NO3

cas num :

616884-63-0

2020 USD :

281

2021 USD :

253 USD

storage :

Store at +4°C

more info or order :

Tocris Bioscience product webpage