UFP-101 | Tocris Bioscience 1552/1 product information

This webpage contains legacy information. The product is either no longer available from the supplier or has been delisted at Labome.

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

UFP-101

catalog :

1552/1

quantity :

1 mg

price :

452 USD

citations: 3

Reference
Wang K, Zheng Y, Yang Y, Wang J, Li B, Wei F, et al. Nociceptin Receptor Is Overexpressed in Non-small Cell Lung Cancer and Predicts Poor Prognosis. Front Oncol. 2019;9:235 pubmed publisher
Mahmoud S, Margas W, Trapella C, Calo G, Ruiz Velasco V. Modulation of silent and constitutively active nociceptin/orphanin FQ receptors by potent receptor antagonists and Na+ ions in rat sympathetic neurons. Mol Pharmacol. 2010;77:804-17 pubmed publisher
Kuzmin A, Sandin J, Terenius L, Ogren S. Evidence in locomotion test for the functional heterogeneity of ORL-1 receptors. Br J Pharmacol. 2004;141:132-40 pubmed

product information

brand :

Tocris, a Bio-Techne Brand

catalog number base :

1552

SKU :

1552/1

product name :

UFP-101

Description :

Potent, selective silent antagonist for NOP

target :

NOP Receptor Antagonists

category :

Peptides

unit size :

1 mg

purity :

95%

observed molecular weight :

1908.19

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=peptides

details of functionality :

UFP-101 is a potent, selective and competitive silent antagonist for the NOP opioid receptor. Binds to NOP with high affinity (pKi = 10.24) and displays 3000-fold selectivity over , u and opioid receptors. Antinociceptive and opposes the action of nociceptin in vivo .

extended description :

Potent, selective silent antagonist for NOP

formula :

C 82 H 138 N 32 O 21

formula text :

C82H138N32O21

cas num :

849024-68-6

USD :

452 USD

product details :

Potent, selective silent antagonist for NOP

alt names :

[Nphe1,Arg14,Lys15]Nociceptin-NH2

storage :

Store at -20°C