GR 231118 | Tocris Bioscience 1486/500 product information

product summary

request information :

company name :

Tocris Bioscience

product type :

chemical

product name :

GR 231118

catalog :

1486/500

quantity :

500µg

price :

329 USD

more info or order :

Tocris Bioscience product webpage

product information

CHEMISTRY :

[H]N[C@@H]([C@@H](C)CC)C(=O)N[C@H]1CCC(=O)NCC(NC(=O)[C@@H]2CCCN2C(=O)[C@H](CCC(=O)NCC(NC(=O)[C@@H]2CCCN2C1=O)C(=O)N[C@@H](CC1=CC=C(O)C=C1)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC1=CC=C(O)C=C1)C(N)=O)NC(=O)[C@@H](N[H])[C@@H](C)CC)C(=O)N[C@@H](CC1=CC=C(O)C=C1)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC1=CC=C(O)C=C1)C(N)=O

Cat Number :

1486/500

Product Name :

GR 231118

Cas Number :

[158859-98-4]

Unit Size :

500µg

Size :

500

Unit :

µg

USD :

329 USD

Primary Category :

7-TM Receptors

Secondary Category :

Peptide Receptors

Tertiary Category :

NPY Receptors

Primary Action :

Potent NPY Y1 antagonist/NPY Y4 agonist. Binds to NPFF receptors

Biological Description :

Potent neuropeptide Y (NPY) Y1 receptor antagonist (pA2 = 10 and 10.5 at rY1 and hY1, receptors respectively). Also a potent and selective NPY Y4 receptor agonist (pEC50 values are 6.0, 8.6 and 6.1 for rY2, hY4 and rY5 receptors respectively). Suppresses food intake in rats in vivo. Also has affinity for neuropeptide FF (NPFF) receptors in vitro (Ki = 43-73 nM).

Formula :

C110H170N34O24

Molwt :

2352.77

Synonyms :

1229U91 GW 1229

more info or order :

Tocris Bioscience product webpage