BMY 14802 hydrochloride | Tocris Bioscience 1440/10 product information

This webpage contains legacy information. The product is either no longer available from the supplier or has been delisted at Labome.

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

BMY 14802 hydrochloride

catalog :

1440/10

quantity :

10 mg (also 50 mg)

price :

149 USD

citations: 2

Reference
Bhide N, Lindenbach D, Surrena M, Goldenberg A, Bishop C, Berger S, et al. The effects of BMY-14802 against L-DOPA- and dopamine agonist-induced dyskinesia in the hemiparkinsonian rat. Psychopharmacology (Berl). 2013;227:533-44 pubmed publisher
Paquette M, Brudney E, Putterman D, Meshul C, Johnson S, Berger S. Sigma ligands, but not N-methyl-D-aspartate antagonists, reduce levodopa-induced dyskinesias. Neuroreport. 2008;19:111-5 pubmed publisher

product information

brand :

Tocris

master code :

1440

SKU :

1440/10

product name :

BMY 14802 hydrochloride

description :

Sigma antagonist. Antipsychotic agent

target :

General Sigma Receptor Antagonists

category :

Small Molecules

sizes available :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

384.86

url print :

?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

BMY 14802 hydrochloride is a potent sigma receptor antagonist (IC50 = 112 nM) with modest to weak affinity for 5-HT1A and 1 receptors. Antipsychotic following oral administration and acts via indirect modulation of central dopaminergic systems.

extended description :

Sigma antagonist. Antipsychotic agent

chemical name text :

-(4-Fluorophenyl)-4-(5-fluoro-2-pyrimidinyl)-1-piperazinebutanol hydrochloride

formula :

C 18 H 22 F 2 N 4 O.HCl

formula text :

C18H22F2N4O.HCl

cas num :

105565-55-7

USD :

141

USD 2023 :

149 USD

product details :

Sigma antagonist. Antipsychotic agent

storage :

Desiccate at RT