SB 228357 | Tocris Bioscience 1375 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

SB 228357

catalog :

1375

quantity :

10 mg (also 50 mg)

price :

153 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

1375

SKU :

1375/10

product name :

SB 228357

description :

5-HT2C/2B antagonist/inverse agonist

target :

5-HT2C Receptor Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

99%

observed molecular weight :

431.39

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

5-HT2C/2B receptor antagonist (pKi values are 7.0, 8.1 and 9.1 at 5-HT2A, 2B and 2C receptors respectively). Displays inverse agonism in a 5-HT-stimulated PI hydrolysis model of 5-HT2C receptor function. Orally active in vivo .

catalog number base :

1375

product keywords :

5-HT2C 5-HT2B antagonists inverse agonists Serotonin Receptors SB228357 5-HT2C Receptors 5-HT2B Receptors 1375,

extended description :

5-HT2C/2B antagonist/inverse agonist

chemical name text :

N-[3-Fluoro-5-(3-pyrindyl)phenyl]-2,3-dihydro-5-methoxy-6-(trifluoromethyl)-1H-indole-1-carboxamide

formula :

C 22 H 17 F 4 N 3 O 2

formula text :

C22H17F4N3O2

cas num :

181629-93-6

2020 USD :

148

2021 USD :

153 USD

storage :

Store at RT

more info or order :

Tocris Bioscience product webpage