chemical

PD 81723

1363

10 mg (also 50 mg)

157 USD

1363

1363/10

PD 81723

Allosteric potentiator of A1 receptors

Adenosine A1 Receptor Modulators

Small Molecules

10 mg (also 50 mg)

99%

299.31

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Allosteric potentiator at the adenosine A1 receptor; acts via agonist-dependent and -independent mechanisms. Enhances agonist affinity for, and increased t of dissociation from, the receptor. Also inhibits basal and forskolin-stimulated adenylyl cyclase (AC) activity in A1 receptors expressed in CHO cells, possibly via direct potentiation of constitutive receptor activity or by direct inhibition of AC. Active in vivo .

1363

Allosteric potentiators A1 receptors Receptors adenosines PD81723 Adenosine A1 Receptors 1363,

Allosteric potentiator of A1 receptors

(2-Amino-4,5-dimethyl-3-thienyl)-[3-(trifluoromethyl)phenyl]methanone

C 14 H 12 F 3 NOS

C14H12F3NOS

132861-87-1

152

157 USD

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