Butabindide oxalate | Tocris Bioscience 1323 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

Butabindide oxalate

catalog :

1323

quantity :

10 mg (also 50 mg)

price :

212 USD

more info or order :

Tocris Bioscience product webpage

citations: 3

Reference
Dasgupta S, Castro L, Dulman R, Yang C, Schmidt M, Ferro E, et al. Proteasome inhibitors alter levels of intracellular peptides in HEK293T and SH-SY5Y cells. PLoS ONE. 2014;9:e103604 pubmed publisher
Lorente E, Garcia R, Lopez D. Allele-dependent processing pathways generate the endogenous human leukocyte antigen (HLA) class I peptide repertoire in transporters associated with antigen processing (TAP)-deficient cells. J Biol Chem. 2011;286:38054-9 pubmed publisher
Duensing S, Darr S, Cuevas R, Melquiot N, Brickner A, Duensing A, et al. Tripeptidyl Peptidase II Is Required for c-MYC-Induced Centriole Overduplication and a Novel Therapeutic Target in c-MYC-Associated Neoplasms. Genes Cancer. 2010;1:883-92 pubmed publisher

product information

brand :

Tocris

master code :

1323

SKU :

1323/10

product name :

Butabindide oxalate

description :

High affinity CCK-inactivating serine protease inhibitor

target :

Additional Synthetic Protease Inhibitors

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

99%

observed molecular weight :

393.44

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

High affinity, reversible, selective and competitive inhibitor of a CCK-inactivating serine protease (tripeptidyl peptidase II) (Ki = 7 nM). Active in vivo (ID50 = 1.1 and 6.8 mg/kg i.v. for inhibition of liver and brain enzyme respectively).

catalog number base :

1323

product keywords :

CCK-inactivating serine protease inhibitors inhibits tripeptidyl peptidase II Proteases Proteinases Cholecystokinin Other Proteases Non-selective CCK 1323,

extended description :

High affinity CCK-inactivating serine protease inhibitor

chemical name text :

(2S)-[1-[(2S)-2-amino-1-oxobutyl]-N-butyl]-2,3-dihydro-1H-indole-2-carboxamide oxalate

formula :

C 17 H 25 N 3 O 2 .C 2 H 2 O 4

formula text :

C17H25N3O2.C2H2O4

cas num :

185213-03-0

2020 USD :

205

2021 USD :

212 USD

storage :

Desiccate at -20°C

more info or order :

Tocris Bioscience product webpage