KT 5823 | Tocris Bioscience 1289/100 product information

product summary

request information :

company name :

Tocris Bioscience

product type :

chemical

product name :

KT 5823

catalog :

1289/100

quantity :

100µg

price :

175 USD

more info or order :

Tocris Bioscience product webpage

product information

CHEMISTRY :

[H][C@]18O[C@](N6C4=C3N1C2=CC=CC=C2C3=C7C(CN(C7=O)C)=C4C5=CC=CC=C56)([C@]([C@@](OC)=O)(OC)C8)C

Cat Number :

1289/100

Product Name :

KT 5823

Cas Number :

[126643-37-6]

Unit Size :

100µg

Size :

100

Unit :

µg

USD :

175 USD

Primary Category :

Enzymes

Secondary Category :

Kinases

Tertiary Category :

Protein Kinase G

Primary Action :

Selective protein kinase G inhibitor

Biological Description :

Selective inhibitor of protein kinase G (Ki values are 0.23, 4 and > 10 μM for inhibition of PKG, PKC and PKA respectively). Inhibits SNP-stimulated PKG activity with an IC50 of 60 nM in dispersed smooth muscle cells and has little effect on PKA activity at concentrations of up to 10 μM.

Formula :

C29H25N3O5

Molwt :

495.53

more info or order :

Tocris Bioscience product webpage