RJR 2429 dihydrochloride | Tocris Bioscience 1271 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

RJR 2429 dihydrochloride

catalog :

1271

quantity :

10 mg (also 50 mg)

price :

163 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

1271

SKU :

1271/10

product name :

RJR 2429 dihydrochloride

description :

nAChR agonist; displays selectivity for 4 2, 1 and 3 4 subtypes

target :

Additional Nicotinic Receptor Agonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

261.19

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent nAChR agonist that displays selectivity for 4 2 (Ki = 1 nM) and 1 subtypes (EC50 values are 297 and 55 nM respectively). Induces dopamine release from striatal neurons (EC50 = 2 nM) and inhibits ion flux in thalamic neurons (IC50 = 154 nM). Also putative 3 4 agonist that potentiates catecholamine release.

catalog number base :

1271

product keywords :

Nicotinic receptor agonists Acetylcholine Receptors Non-Selective Subtypes nAChR RJR2429 dihydrochloride Nicotinic Receptors (Non-selective) 1271,

extended description :

nAChR agonist; displays selectivity for 4 2, 1 and 3 4 subtypes

chemical name text :

( )-2-(3-Pyridinyl)-1-azabicyclo[2.2.2]octane dihydrochloride

formula :

C 12 H 16 N 2 .2HCl

formula text :

C12H16N2.2HCl

cas num :

1021418-53-0

2020 USD :

159

2021 USD :

163 USD

storage :

Desiccate at RT

more info or order :

Tocris Bioscience product webpage