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company name :
Tocris Bioscience
product type :
chemical
product name :
1268/10
catalog :
1268/10
quantity :
10 mg (also 50 mg)
price :
207 USD
more info or order :
citations: 93
Reference
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product information
master code :
1268
SKU :
1268/10
product name :
U 73122
unit size :
10 mg (also 50 mg)
description :
Phospholipase C inhibitor
target :
Phospholipase Inhibitors
category :
Small Molecules
purity :
98%
observed molecular weight :
464.65
url print :
?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules
details of functionality :
U 73122 is a phospholipase C inhibitor. Inhibits agonist-induced platelet aggregation with IC50 values of 1-5 u M. Potently inhibits human polymorphonuclear neutrophil adhesion on biological surfaces (IC50 50 nM) and exhibits antinociceptive activity in vivo . Also activates TRPM4 and inhibits TRPM3 channels. . Negative Control also available.
top caption :
Phospholipase C inhibitor
extended description :
Phospholipase C inhibitor
chemical name text :
1-[6-[[(17 )-3-Methoxyestra-1,3,5(10)-trien-17-yl]amino]hexyl]-1H-pyrrole-2,5-dione
formula :
C29H40N2O3
formula text :
C29H40N2O3
cas num :
112648-68-7
USD :
207 USD
product details :
Phospholipase C inhibitor
storage :
Store at RT
more info or order :
company information
Tocris Bioscience
The Watkins Building
Atlantic Road
Avonmouth, Bristol
BS11 9QD
info@bio-techne.com
https://www.tocris.com
800-343-7475
headquarters: UK