FR 139317 | Tocris Bioscience 1210/10 product information

This webpage contains legacy information. The product is either no longer available from the supplier or has been delisted at Labome.

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

FR 139317

catalog :

1210/10

quantity :

10 mg (also 50 mg)

price :

271 USD

citations: 1

Reference
Khodorova A, Richter J, Vasko M, Strichartz G. Early and late contributions of glutamate and CGRP to mechanical sensitization by endothelin-1. J Pain. 2009;10:740-9 pubmed publisher

product information

brand :

Tocris

master code :

1210

SKU :

1210/10

product name :

FR 139317

description :

Highly potent, selective ETA antagonist

target :

Endothelin ETA Receptor Antagonists

category :

Small Molecules

sizes available :

10 mg (also 50 mg)

purity :

99%

observed molecular weight :

604.75

url print :

?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

FR 139317 is a highly potent and selective ETA endothelin receptor antagonist (Ki values are 1 nM and 7.3 u M at ETA and ETB subtypes respectively). Active in vivo .

extended description :

Highly potent, selective ETA antagonist

chemical name text :

N-[N-[N-[(Hexahydro-1H-azepin-1-yl)carbonyl]-L-leucyl]-1-methyl-D-tryptophyl]-3-(2-pyridinyl)-D-alanine

formula :

C 33 H 44 N 6 O 5

formula text :

C33H44N6O5

cas num :

142375-60-8

USD :

258

USD 2023 :

271 USD

product details :

Highly potent, selective ETA antagonist

storage :

Desiccate at +4°C